Inhibitors/Activators

Small molecule enzyme inhibitors and activators are compounds that can modulate the activity of enzymes. Enzyme inhibitors bind to enzymes and prevent them from catalyzing reactions, while enzyme activators enhance their catalytic activity. Small molecules have significant therapeutic potential, providing some pharmacological advantages over biologics and are used in treating diseases caused by overactive or underactive enzymes or targeting pathogen-specific enzymes. Enzyme inhibitors and activators remain an active area of research in drug discovery and development. BPS Bioscience provides known positive controls for inhibitors and activators to affect protein function or for use in our biochemical and cell-based assays.
Molecular model of SARS-CoV-2 3CL

Molecular model of SARS-CoV-2 3CL protease dimer (teal/blue) in complex with inhibitor GC376 based on PDB ID 7CBT.

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437 total products

Displaying 25 products per page

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Catalog #
Name
Size
Target Category
Protein Target(s)
Function
KY 2111
50 mg
Wnt Signaling
 
Inhibitor
KY 2111
200 mg
Wnt Signaling
 
Inhibitor
KY 2111
10 mg
Wnt Signaling
 
Inhibitor
Posaconazole
25 mg
Demethylases
14α-demethylase
Inhibitor
Posaconazole
5 mg
Demethylases
14α-demethylase
Inhibitor
Lactacystin
500 µg
Ubiquitin
20S Proteasome
Inhibitor
PS-341 (MG-341)
5 mg
Ubiquitin
20S Proteasome
Inhibitor
PS-341 (MG-341)
25 mg
Ubiquitin
20S Proteasome
Inhibitor
DBeQ
25 mg
Ubiquitin
AAA-ATPase p97
Inhibitor
DBeQ
10 mg
Ubiquitin
AAA-ATPase p97
Inhibitor
Vismodegib (GDC-04491)
25 mg
Miscellaneous
ABCG2/BCRP, ABCB1/Pgp
Inhibitor
Vismodegib (GDC-04491)
50 mg
Miscellaneous
ABCG2/BCRP, ABCB1/Pgp
Inhibitor
ND-630
1 mg
Metabolic Enzymes
ACC1, ACC2
Inhibitor
ND-630
5 mg
Metabolic Enzymes
ACC1, ACC2
Inhibitor
Donepezil HCl
5 g
Metabolism
AChE
Inhibitor
Donepezil HCl
1 g
Metabolism
AChE
Inhibitor
Forskolin
100 mg
cAMP/kinase
Adenylyl cyclase
Activator
Forskolin
50 mg
cAMP/kinase
Adenylyl cyclase
Activator
AICAR
25 mg
ACC
AMPK
Activator
A-769662
10 mg
Kinases
AMPK
Activator
TAME-HCL
100 mg
Ubiquitin
APC/C
Inhibitor
(S)-MG132
10 mg
Ubiquitin
B16, IPC227F
Inhibitor
BAM7
50 mg
Apoptosis
BAX
Activator
BAM7
10 mg
Apoptosis
BAX
Activator
Obatoclax
5 mg
Apoptosis
Bcl-2
Inhibitor