Telotristat
Catalog #
27341
$425
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Description
Telotristat is the active metabolite of LX1606 (Telotristat etiprate), which is an orally bioavailable, small-molecule, tryptophan hydroxylase (TPH) inhibitor with potential antiserotonergic activity.
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Synonyms
LX1032
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Product Data Gallery
Product Info
Storage and Usage
Citations
Purity
≥98%
Formula
C25H22CIF3N6O3
MW
547 Da
Solubility
Soluble in DMSO (10 mM). Only sparingly soluble in water (<1.5 µg/ml).
Biological Activity
Telotristat has been reported to inhibit the TPH enzyme. This inhibition can reduce serotonin production in the periphery.
CAS Registry #
1033805-28-5
References
1. Kulke, M., et al., Endocr. Relat. Cancer, 2014; 21: 705-714.
2. Margolis, K.G. et al., Gut, 2014; 63(6):928-37.
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