Telotristat

Catalog #

27340

$255 *

Size: 5 mg

Qty

Bulk/Custom

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Description

Telotristat is the active metabolite of LX1606 (Telotristat etiprate), which is an orally bioavailable, small-molecule, tryptophan hydroxylase (TPH) inhibitor with potential antiserotonergic activity.

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Synonyms

LX1032

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Product Data Gallery

Product Info

Storage and Usage

Citations

Purity

≥98%

Format

White powder

Formula

C₂₅H₂₂CIF₃N₆O₃

546.93 Da

Solubility

≥27.35 mg/mL in DMSO with ultrasonic; insoluble in H2O; insoluble in EtOH

Biological Activity

Telotristat has been reported to inhibit the TPH enzyme. This inhibition can reduce serotonin production in the periphery.

CAS Registry #

1033805-28-5

References

1. Kulke, M., et al., Endocr. Relat. Cancer, 2014; 21: 705-714.

2. Margolis, K.G. et al., Gut, 2014; 63(6):928-37.

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Telotristat

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