GSK-6853

Catalog #

82067

$525 *

Size: 50 mg

Qty

Bulk/Custom

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*US Pricing only. For international pricing, please contact your local distributor.

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Description

GSK-6853 is a potent and selective BRPF1 inhibitor. GSK-6853 exhibits >1600-fold selectivity for BRPF1 over other bromodomains (pIC₅₀ values by TR-FRET are 8.1, 5.1/4.8 and 4.7/<4.3 for BRPF1, BRPF2/3 and BRD4 BD1/2, respectively). The structural analog of GSK-6853, GSK-9311, serves as a good inactive control (125- and 185-fold reduced potency in cell-free and cell-based assays, respectively).

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Synonyms

GSK6853, GSK 6853

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