GSK-5959

Catalog #

82066

$330 *

Size: 25 mg

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Bulk/Custom

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Description

GSK-5959 exhibits >100-fold selectivity for BRPF1 (IC₅₀ = 80 nM) over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3, which is involved in the epigenetic regulation of gene expression and have been implicated in human cancer.

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Synonyms

GSK5959, GSK 5959

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